首页> 外国专利> SOLID PHARMACEUTICAL COMPOSITION ADMINISTRATIBLE ORALLY, USE OF THE PHARMACEUTICAL COMPOSITION, PROCESS FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS, AND METHOD OF TREATING A PATIENT SUFFERING FROM PATHOLOGICAL CONDITIONS

SOLID PHARMACEUTICAL COMPOSITION ADMINISTRATIBLE ORALLY, USE OF THE PHARMACEUTICAL COMPOSITION, PROCESS FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS, AND METHOD OF TREATING A PATIENT SUFFERING FROM PATHOLOGICAL CONDITIONS

机译:固体药品成分可管理的口服制剂,药品成分的使用,药品成分的制备过程以及治疗患者的病理状况的方法

摘要

the invention relates to oral pharmaceutical compositions for the administration of modified release of cariprazine (trans-n- {4- [2- [4- (2,3-dichlorophenyl) -piperazin-1-yl] -ethyl] -cycle -hexyl} -n?, n? -dimethylurea) or pharmaceutically acceptable salts thereof, for dosage less than daily. the invention also relates to the use of said compositions in the treatment and / or prevention of pathological conditions that require modulation of dopamine receptors. the invention also relates to the process for preparing said modified release pharmaceutical compositions.
机译:本发明涉及口服施用的药物组合物,该药物组合物用于给予卡比拉嗪(反式-n- {4- [2- [2-(4-(2,3-二氯苯基)-哌嗪-1-基]-乙基])-环-己基-n′,n′-二甲基脲)或其药学上可接受的盐,其剂量少于每日一次。本发明还涉及所述组合物在治疗和/或预防需要调节多巴胺受体的病理状况中的用途。本发明还涉及制备所述调释药物组合物的方法。

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