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NEW PHOSPHANICAL AND ASPHOSPHANIAN PRODUCTS, METHOD OF ADMINISTRATION AND PHARMACEUTICAL SUBSTANCES CONTAINING THEM

机译:新型农药和农药产品,包含其的管理方法和药物

摘要

Compounds of type (I) where: Ak1 is an alkyl solution,X represents -(CH2)m-,-CH(R)-,N(R)-,-CH2-N(R)-,-N(R)-CH2- or -CH2-N(R)-CH2-,m and R are as defined in the description,R1 and R2 each represent H when X represents -(CH2)m-,-CH(R)-,N(R)-CH2-N(R)- or -N(R)-CH2- or indeed together form a bond when X represents -CH2-N(R)-CH2-,R3 represents NH2, Cy-NH2, Cy-Ak3-NH2 or piperidine-4-yl,Cy and Ak3 are as defined in the description,R4 and R5, identical or different,Each represents H or F, their optical isomers and their medically acceptable salts of added acid. The invention also applies to medicines containing them.
机译:类型(I)的化合物,其中:Ak1是烷基溶液,X表示-(CH2)m-,-CH(R)-,N(R)-,-CH2-N(R)-,-N(R) -CH 2-或-CH 2 -N(R)-CH 2-,m和R如说明书中所定义,当X表示-(CH 2)m-,-CH(R)-,N(-时,R 1和R 2各自代表H。 R)-CH2-N(R)-或-N(R)-CH2-或实际上一起形成键,当X代表-CH2-N(R)-CH2-时,R3代表NH2,Cy-NH2,Cy-Ak3 -NH 2或哌啶-4-基,C y和Ak 3如说明书中所定义,R 4和R 5相同或不同,每个代表H或F,它们的旋光异构体和其医学上可接受的加成盐。本发明也适用于含有它们的药物。

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