首页> 外国专利> NOVEL PYRIDO3,4-DPYRIMIDIN-8-ONE DERIVATIVE HAVING PROTEIN KINASE INHIBITORY ACTIVITY, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING, ALLEVIATING, OR TREATING CANCER, COMPRISING SAME

NOVEL PYRIDO3,4-DPYRIMIDIN-8-ONE DERIVATIVE HAVING PROTEIN KINASE INHIBITORY ACTIVITY, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING, ALLEVIATING, OR TREATING CANCER, COMPRISING SAME

机译:新型PYRIDO [3,4-D] PYRIMIDIN-8衍生物具有蛋白激酶抑制活性,以及​​用于预防,转移或治疗癌症的药物组合物,包括相同的成分

摘要

The present invention relates to: a pyrido[3,4-d]pyrimidin-8-one derivative compound exhibiting excellent anti-proliferative effects on cancer cells, a pharmaceutically acceptable salt thereof, a hydrate thereof, or a stereoisomer thereof; a preparation method therefor; a pharmaceutical composition for preventing, alleviating, or treating cancer metastasis and proliferative diseases, containing same as an active ingredient; and an anti-cancer composition used on cancer cells, wherein the compound exhibits excellent cancer cell inhibitory activities and anti-proliferative effects, thereby being useful in the inhibition of cancer cells and, further, in the prevention of cancer metastasis and proliferative diseases and in the cancer treatment.
机译:本发明涉及一种对癌细胞具有优异的抗增殖作用的吡啶并[3,4-d]嘧啶-8-衍生物化合物,其药学上可接受的盐,其水合物或立体异构体。其制备方法;用于预防,减轻或治疗癌症转移和增生性疾病的药物组合物,含有该药物组合物作为活性成分;以及用于癌细胞的抗癌组合物,其中所述化合物表现出优异的癌细胞抑制活性和抗增殖作用,从而可用于抑制癌细胞,并且进一步用于预防癌症转移和增生性疾病以及用于治疗癌症。癌症治疗。

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