;EFFECT: said compound is suitable as an ATR protein kinase inhibitor.;10 cl, 9 dwg, 6 tbl, 8 ex"/> RADIOLABELLED 2-AMINO-6-FLUORO-N-5-FLUORO-PYRIDIN-3-YL-PYRAZOLO 1, 5-A PYRIMIDINE-3-CARBOXAMIDE DERIVATIVES USED AS ATR KINASE INHIBITOR, PREPARATIONS BASED THEREON COMPOUNDS AND VARIOUS SOLID FORMS THEREOF
首页> 外国专利> RADIOLABELLED 2-AMINO-6-FLUORO-N-5-FLUORO-PYRIDIN-3-YL-PYRAZOLO 1, 5-A PYRIMIDINE-3-CARBOXAMIDE DERIVATIVES USED AS ATR KINASE INHIBITOR, PREPARATIONS BASED THEREON COMPOUNDS AND VARIOUS SOLID FORMS THEREOF

RADIOLABELLED 2-AMINO-6-FLUORO-N-5-FLUORO-PYRIDIN-3-YL-PYRAZOLO 1, 5-A PYRIMIDINE-3-CARBOXAMIDE DERIVATIVES USED AS ATR KINASE INHIBITOR, PREPARATIONS BASED THEREON COMPOUNDS AND VARIOUS SOLID FORMS THEREOF

机译:放射性标记的2-氨基-6-氟-N- [5-氟-吡啶-3-基]-吡唑啉[1,5-A]嘧啶-3-甲酰胺衍生物用作抗逆转录酶激酶抑制剂,基于其化合物和各种固体的制备形式

摘要

FIELD: chemistry.;SUBSTANCE: present invention relates to a method of producing a compound of formula I-1, which includes a step of reacting a compound of formula 6b with a compound of formula 11. ; ;EFFECT: said compound is suitable as an ATR protein kinase inhibitor.;10 cl, 9 dwg, 6 tbl, 8 ex
机译:式I-1化合物的制备方法技术领域本发明涉及式I-1的化合物的制备方法,其包括使式6b的化合物与式11的化合物反应的步骤。 效果:所述化合物适合作为ATR蛋白激酶抑制剂。; 10 cl,9 dwg,6 tbl,8 ex

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