N- and S-alpha-l-arabinopyranosyl(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazoles. First synthesis and biological evaluation.

Khalil NS

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N- and S-alpha-l-arabinopyranosyl(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazoles. First synthesis and biological evaluation.

机译：N-和S-α-1-阿拉伯吡喃并（1,2,4）三唑（3,4-b）（1,3,4）噻二唑。首先进行合成和生物学评估。

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摘要

First synthesis of N- and S-alpha-l-arabinopyranosyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles is described. Antimicrobial screening of two selected regioisomeric compounds against Aspergillus fumigatus, Penicillium italicum, Syncephalastrum racemosum, Candida albicans, Staphylococcus aureus, Pseudomonas aeruginosa, Bacillus subtilis and Escherichia coli are compared.

机译：描述了N-和S-α-1-阿拉伯吡喃糖基[1,2,4]三唑并[3,4-b] [1,3,4]噻二唑的首次合成。比较了针对烟曲霉，意大利青霉菌，总青霉，白念珠菌，金黄色葡萄球菌，铜绿假单胞菌，枯草芽孢杆菌和大肠杆菌的两种选定的区域异构化合物的抗菌筛选。

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《European Journal of Medicinal Chemistry: Chimie Therapeutique》 |2007年第9期|共7页
作者
Khalil NS;
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正文语种 eng
中图分类医药、卫生;劳动卫生;
关键词
Anti-Infective Agents; Bacteria; Drug Evaluation; Preclinical; Fungi; Magnetic Resonance Spectroscopy; 抗感染药; 细菌; 真菌; 微生物敏感性试验; 噻二唑类;

机译：Anti-Infective Agents;Bacteria;Drug Evaluation;Preclinical;Fungi;Magnetic Resonance Spectroscopy;抗感染药;细菌;真菌;微生物敏感性试验;噻二唑类;

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1. N- and S-alpha-l-arabinopyranosyl(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazoles. First synthesis and biological evaluation. [J] . Khalil NS European Journal of Medicinal Chemistry: Chimie Therapeutique . 2007,第9期

机译：N-和S-α-1-阿拉伯吡喃并（1,2,4）三唑（3,4-b）（1,3,4）噻二唑。首先进行合成和生物学评估。
2. Novel simple efficient synthetic approach toward 6-substituted-2H-(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazole-3-thiones and first synthesis and biological evaluation of N-and S-beta-D-glucosides of the(1,2,4)triazolo (3,4-b)(1,3,4)thiadiazole ring syste [J] . Khalil NS Nucleosides, nucleotides and nucleic acids . 2007,第4期

机译：一种新的简单有效的合成方法，用于6-取代的2H-（1,2,4）三唑并（3,4-b）（1,3,4）噻二唑-3-硫酮和N-和S的首次合成和生物学评价（1,2,4）三唑（3,4-b）（1,3,4）噻二唑环系的-β-D-葡萄糖苷
3. Convenient synthesis of some 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines bearing 3-methylthio{7H-1,2,4-triazolo[1,5-d]tetrazol-6-yl}moiety as possible antimicrobial activity [J] . Taha MAM Phosphorus, Sulfur, and Silicon and the Related Elements . 2008,第10期

机译：方便合成一些1,2,4-三唑并[3,4-b] -1,3,4-噻二唑和1,2,4-三唑并[3,4-b] -1,3,4-噻二嗪3-甲硫基{7H-1,2,4-三唑并[1,5-d]四唑-6-基}部分尽可能具有抗菌活性
4. A New Method for the Synthesis of Novel S-Triazolo3,4-b 1,3,4Thiadiazines [C] . Sattar Ebrahimi, Naser Foroughifar, Akbar Mobinikhaledi European Symposium on Organic Chemistry . 2009

机译：新型S-Tri唑的合成方法3,4-B 1,3,4噻二嗪
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机译：第一部分。天然激素α，25-二羟基维生素D（3）的新型类似物：设计，合成和生物学评估。第二部分n尺寸的2-环烯酮新的硅介导的环扩展成中等烯丙基n + 3和羟基烯属n + 3 + m中等尺寸的内酯：（+）-顺-月桂聚糖和（-）-紫杉醇-J的全合成。
6. 6-(4-Bromophenyl)-3-methyl-7H-1,2,4-triazolo[3,4-b][1,3,4]thiadiazine [O] . Hoong-Kun Fun, Ching Kheng Quah, Hatem A. Abdel-Aziz, 2015

机译：6-（4-溴基）-3-甲基-7H-1,2,4-三唑[3,4-b] [1,3,4]噻二嗪
7. Synthesis and antiviral activity of novel [1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles, [1,2,4]triazolo[3,4-b] [1,3,4]thiadiazines and [1,2,4]triazolo[3,4-b][1,3,4] thiadiazepines [O] . Abdel-Rahman Farghaly, Erik De Clercq, Hussein El-Kashef 2006

机译：新[1,2,4]三唑并[3,4-b] [1,3,4]噻二唑，[1,2,4]三唑并[3,4-b] [1,3]的合成及抗病毒活性4]噻二嗪和[1,2,4]三唑并[3,4-b] [1,3,4]噻二氮杂

N- and S-alpha-l-arabinopyranosyl(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazoles. First synthesis and biological evaluation.

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