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机译:聚合物载体和棕榈酸 - 缀合的siRNA之间的疏水相互作用改善了聚乙二醇化的多重稳定性,增强了体内药代动力学和肿瘤基因沉默
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
Vanderbilt Univ Vanderbilt Inst Nanoscale Sci &
Engn Dept Biomed Engn Sch Engn Nashville TN;
RNA interference; PEGylated polyplexes; Pharmacokinetics; Hydrophobicity; Breast cancer; Tumor targeting;
机译:聚合物载体和棕榈酸 - 缀合的siRNA之间的疏水相互作用改善了聚乙二醇化的多重稳定性,增强了体内药代动力学和肿瘤基因沉默
机译:PEG架构和疏水含量的组合优化改善了三元患者型多重稳定性,药代动力学和体内效力
机译:棕榈酸缀合的21个核苷酸siRNA可增强基因沉默活性。
机译:优化PEG长度以增强胶束siRNA载体的体内药代动力学
机译:固定化细胞色素P450 2C9(CYP2C9):用于代谢物生成,监测蛋白质-蛋白质相互作用以及使用增强的体外模型改善体内预测的应用
机译:高分子载体与棕榈酸缀合的siRNA之间的疏水相互作用可改善PEG化多态复合物的稳定性并增强体内药代动力学和肿瘤基因沉默。
机译:聚乙二醇化多态胶束在肿瘤缺氧中的增强渗滤和基因表达