机译:基于苄胺的配体的发现与设计与补体因子D解锁构象的结合
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Novartis Pharma AG Institutes for BioMedical Research Novartis Campus CH-4056 Basel Switzerland;
Alternative complement pathway; factor D inhibitors; fragment-based drug discovery; structure-based design;
机译:基于苄胺的配体的发现与设计与补体因子D解锁构象的结合
机译:基于吡咯烷的β-分泌酶抑制剂的发现:通过构象设计提高铅的水平,以维持配体结合效率
机译:CDK8 / CYC和配体结合的分子动力学研究:组织柔韧性和药物发现中的含义
机译:使用羟基自由基足迹对CCL5-chondrotin硫酸盐复合物的研究显示涉及配体结合,配体诱导的构象变化和pH依赖聚集的信息
机译:六聚体胰岛素HisB10结合位点的羧酸盐配体的设计,合成和定量结构活性关系,以及使用动态核磁共振(DNMR)光谱法检测酚类配体的结合机理。
机译:第一种基于苄胺的配体的发现和设计绑定到补体因子D的解锁构象
机译:基于苄胺基配体的发现与设计与补体因子D解锁构象的结合