机译:RETV804M激酶的WT-RET / KDR选择性抑制剂的发现与优化
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Univ Leicester Dept Mol &
Cell Biol Henry Wellcome Bldg Leicester LE1 7RH Leics England;
Univ Leicester Dept Mol &
Cell Biol Henry Wellcome Bldg Leicester LE1 7RH Leics England;
Univ Leeds Fac Biol Sci Astbury Ctr Struct Mol Biol Leeds LS2 9JT W Yorkshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Univ Leicester Dept Mol &
Cell Biol Henry Wellcome Bldg Leicester LE1 7RH Leics England;
Univ Leeds Fac Biol Sci Astbury Ctr Struct Mol Biol Leeds LS2 9JT W Yorkshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
Canc Res Drug Discovery Unit Macclesfield Cheshire England;
RET; KDR; kinase inhibitor; virtual screening;
机译:RETV804M激酶的WT-RET / KDR选择性抑制剂的发现与优化
机译:丝裂素活化的蛋白激酶活化的蛋白激酶2(MAPKAP-K2)作为抗炎目标:使用聚焦库和基于结构的优化方法,发现选择性吡唑并[1,5-a]嘧啶抑制剂并具有体内活性
机译:二氢吡咯并吡唑系列转化生长因子-βI型受体激酶域抑制剂的优化:口服生物利用转化生长因子-β受体I型抑制剂作为抗肿瘤药的发现
机译:探索蛋白酪氨酸激酶抑制剂发现中离子迁移率质谱的潜力
机译:计算机辅助发现的受体酪氨酸激酶的新型天然产物抑制剂及其对多种恶性肿瘤的合理的半合成优化。
机译:大环喹喔啉-吡咯并-二氢哌啶子酮的发现和优化作为有效的Pim-1 / 2激酶抑制剂
机译:校正“发现和优化4,5-二芳基氧唑作为丙酮酸脱氢酶激酶和热休克蛋白90的有效双重抑制剂”