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机译:铬酮衍生物作为多功能支架,具有双向抑制HIV-1逆转录酶相关的核糖核酸酶H函数和整合酶活性
Univ Cagliari Dept Life &
Environm Sci Cittadella Univ SS554 I-09042 Monserrato CA Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Dept Life &
Environm Sci Via Osped 72 I-09124 Cagliari Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Dept Life &
Environm Sci Via Osped 72 I-09124 Cagliari Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Magna Graecia Univ Catanzaro Net4Sci Acedem Spin Off Campus S Venuta Viale Europa I-88100;
Alexander Educ Inst Thessaloniki Sch Hlth &
Med Care Dept Med Lab Studies Sindos Greece;
Potel JDK Davolwala Sci Coll Dept Chem Anand Gujarat India;
Alexander Educ Inst Thessaloniki Sch Hlth &
Med Care Dept Med Lab Studies Sindos Greece;
Potel JDK Davolwala Sci Coll Dept Chem Anand Gujarat India;
Potel JDK Davolwala Sci Coll Dept Chem Anand Gujarat India;
Univ Cagliari Dept Life &
Environm Sci Cittadella Univ SS554 I-09042 Monserrato CA Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Magna Graecia Univ Catanzaro Dept Hlth Sci Campus S Venuta Viale Europa I-88100 Catanzaro Italy;
Aristotle Univ Thessaloniki Sch Pharm Dept Med Chem Thessaloniki Greece;
Univ Cagliari Dept Life &
Environm Sci Cittadella Univ SS554 I-09042 Monserrato CA Italy;
Coumarin derivatives; HIV-1; RNase H; Integrase; Dual inhibitors; LEDGF/p75 cellular cofactor;
机译:铬酮衍生物作为多功能支架,具有双向抑制HIV-1逆转录酶相关的核糖核酸酶H函数和整合酶活性
机译:过去和未来。当前针对HIV-1整合酶和逆转录酶相关的核糖核酸酶H活性的药物:单和双活性位点抑制剂。
机译:预测双靶吡咯基Diketo酸支架对HIV-1整合酶和反转录酶相关核糖核酸酶H的结合模式和电阻曲线
机译:喹啉酸衍生物作为HIV-1整合酶抑制的喹啉酸衍生物的合成与生物学评价
机译:HIV-1整合酶抑制的新模式
机译:支架跳跃和优化34-二羟基苯基 - 含硫基嘧啶酮:喹唑啉酮衍生物的合成作为HIV-1逆转录酶相关核糖核酸酶H的新型变形抑制剂
机译:羟基化的对苯二酚选择性抑制HIV-1逆转录酶相关的核糖核酸酶H的活性