One-pot synthesis of arylated 1-methyl-1H-indoles by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H-indole

Ibad M.F.; Zinad D.S.; Hussain M.; Ali A.; Villinger A.; Langer P.

首页> 外文期刊>Tetrahedron >One-pot synthesis of arylated 1-methyl-1H-indoles by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H-indole

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One-pot synthesis of arylated 1-methyl-1H-indoles by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H-indole

机译：通过2,3-二溴-1-甲基-1H-吲哚和2,3,6-三溴-1-甲基-1H-的Suzuki-Miyaura交叉偶联反应一锅合成芳基化的1-甲基-1H-吲哚吲哚

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Arylated 1-methyl-1H-indoles were prepared by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H- indole. The reactions proceed with very good regioselectivity in favour of position 2.

机译：通过Suzuki-Miyaura的2,3-二溴-1-甲基-1H-吲哚和2,3,6-三溴-1-甲基-1H-吲哚的Suzuki-Miyaura交叉偶联反应，制备了丙烯酸化的1-甲基-1H-吲哚。反应以非常好的区域选择性进行，有利于位置2。

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《Tetrahedron》 |2013年第35期|共13页
作者
Ibad M.F.; Zinad D.S.; Hussain M.; Ali A.; Villinger A.; Langer P.;
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正文语种 eng
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关键词
Catalysis; Cross-coupling; N-Heterocycles; Palladium; Suzuki-Miyaura reaction;

机译：催化;交叉偶联;N-杂环;钯;Suzuki-Miyaura反应;

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1. One-pot synthesis of arylated 1-methyl-1H-indoles by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H-indole [J] . Ibad M.F., Zinad D.S., Hussain M., Tetrahedron . 2013,第35期

机译：通过2,3-二溴-1-甲基-1H-吲哚和2,3,6-三溴-1-甲基-1H-的Suzuki-Miyaura交叉偶联反应一锅合成芳基化的1-甲基-1H-吲哚吲哚
2. Efficient synthesis of arylated flavones by site-selective Suzuki-Miyaura cross-coupling reactions of the bis(triflate) of 5,7- and 7,8-dihydroxyflavone [J] . Eleya N., Malik I., Reimann S., European journal of organic chemistry . 2012,第8期

机译：通过5,7-和7,8-二羟基黄酮双（三氟甲磺酸酯）的位点选择性Suzuki-Miyaura交叉偶联反应有效合成芳基化黄酮
3. Efficient Synthesis of Arylated Coumarins by Site-Selective Suzuki-Miyaura Cross-Coupling Reactions of the Bis(tritlate) of 4-Methy1-5,7-dihydroxy coumarin [J] . Nadi Eleya, Zein Khaddour, Tunas Patonay, Synlett . 2012,第2期

机译：4-位甲基1-5,7-二羟基香豆素的双（三氟甲磺酸盐）的位点选择性Suzuki-Miyaura交叉偶联反应有效合成丙烯酸化的香豆素
4. Rationalizing the selectivity of the Suzuki-Miyaura cross-coupling reaction in the synthesis of 1-arylnaphthalenes and 1,8-diarylnaphthalenes. [C] . Carlos F. R. A. C. Lima, Luis M. N. B. F. Santos, Jose E. Rodriguez-Borges European Symposium on Organic Chemistry . 2009

机译：合理化Suzuki-Miyaura交叉偶联反应在合成1-芳基萘和1,8-二芳基萘中的选择性。
5. Design, synthesis and Suzuki-Miyaura cross-coupling reactions of potassium organotrifluoroborates. [D] . Shin, Inji. 2013

机译：有机三氟硼酸钾的设计，合成和Suzuki-Miyaura交叉偶联反应。
6. Direct One-Pot Synthesis of Primary 4-Amino-23-diaryl- quinolines via Suzuki-Miyaura Cross-Coupling of 2-Aryl-4-azido-3-iodoquinolines with Arylboronic Acids [O] . Malose Jack Mphahlele, Mamasegare Mabel Mphahlele 2011

机译：通过2-芳基-4-叠氮基-3-碘喹啉与芳基硼酸的铃木-宫浦交叉偶合直接一锅合成伯4-氨基-23-二芳基-喹啉
7. Suzuki-Miyaura Reactions of Arenediazonium Salts Catalyzed by Pd(0)/C. One-Pot Chemoselective Double Cross-Coupling Reactions [O] . -1

机译：Suzuki-miyaura通过Pd（0）/ c催化的氧化亚氮盐的反应。单壶化学选择双交叉偶联反应

One-pot synthesis of arylated 1-methyl-1H-indoles by Suzuki-Miyaura cross-coupling reactions of 2,3-dibromo-1-methyl-1H-indole and 2,3,6-tribromo-1-methyl-1H-indole

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