AN EXPEDIENT ONE-POT SYNTHESIS FOR PROTECTED 2-THIA-5-AZABICYCLO[2.2.1]HEPTAN-3-ONES - VERSATILE INTERMEDIATES IN THE SYNTHESIS OF CARBAPENEM SIDECHAINS

Brands KMJ.; Williams JM.; Dolling UH.; Reider PJ.; Marchesini G.

首页> 外文期刊>Tetrahedron letters: The International Journal for the Rapid Publication of Preliminary Communications in Organic Chemistry >AN EXPEDIENT ONE-POT SYNTHESIS FOR PROTECTED 2-THIA-5-AZABICYCLO[2.2.1]HEPTAN-3-ONES - VERSATILE INTERMEDIATES IN THE SYNTHESIS OF CARBAPENEM SIDECHAINS

【24h】

AN EXPEDIENT ONE-POT SYNTHESIS FOR PROTECTED 2-THIA-5-AZABICYCLO[2.2.1]HEPTAN-3-ONES - VERSATILE INTERMEDIATES IN THE SYNTHESIS OF CARBAPENEM SIDECHAINS

机译：受保护的2-thia-5-azabicyclo [2.2.1] Heptan-3-ones的一种便捷的一锅合成方法，该中间体在卡宾木苷的合成中

获取原文

获取原文并翻译 | 示例

掌桥外文数据库（机构版） >>

开具论文收录证明 >>

文献代查 >>

页面导航

摘要
著录项
相似文献
相关主题

摘要

A convenient and high yielding one-pot process for the preparation of protected 2-thia-5-azabicyclo-[2.2.1]heptan-3-ones from 4-hydroxyproline and their use in the synthesis of carbapenem sidechains is described. (C) 1996 Elsevier Science Ltd [References: 12]

机译：描述了一种方便且高产率的一锅法，用于从4-羟基脯氨酸制备受保护的2-thia-5-azabicyclo- [2.2.1]庚烷-3-酮及其在碳青霉烯侧链合成中的应用。（C）1996 Elsevier Science Ltd [参考：12]

著录项

来源
《Tetrahedron letters: The International Journal for the Rapid Publication of Preliminary Communications in Organic Chemistry》 |1996年第17期|共4页
作者
Brands KMJ.; Williams JM.; Dolling UH.; Reider PJ.; Marchesini G.;
展开▼
作者单位

展开▼
收录信息
原文格式 PDF
正文语种 eng
中图分类有机化学;
关键词

相似文献

外文文献
中文文献
专利

1. AN EXPEDIENT ONE-POT SYNTHESIS FOR PROTECTED 2-THIA-5-AZABICYCLO[2.2.1]HEPTAN-3-ONES - VERSATILE INTERMEDIATES IN THE SYNTHESIS OF CARBAPENEM SIDECHAINS [J] . Brands KMJ., Williams JM., Dolling UH., Tetrahedron letters: The International Journal for the Rapid Publication of Preliminary Communications in Organic Chemistry . 1996,第17期

机译：受保护的2-thia-5-azabicyclo [2.2.1] Heptan-3-ones的一种便捷的一锅合成方法，该中间体在卡宾木苷的合成中
2. SYNTHESIS OF (+)- AND (-)-N-BOC-7-AZABICYCLO[2.2.1]HEPTAN-2-ONES VERSATILE INTERMEDIATES FOR THE ENANTIOSPECIFIC SYNTHESIS OF (+)- AND (-)-EPIBATIDINE AND ANALOGUES [J] . Hernandez A., Rapoport H., Marcos M. The Journal of Organic Chemistry . 1995,第9期

机译：（+）-和（-）-N-BOC-7-氮杂双环[2.2.1] Heptan-2-one多功能中间体的合成（+）-和（-）-表皮苷和类似物的对映体
3. Design and synthesis of m1-selective muscarinic agonists: (R)-(-)-(Z)-1-Azabicyclo(2.2.1)heptan-3-one, O-(3-(3'-methoxyphenyl)-2-propynyl)oxime maleate (CI-1017), a functionally m1-selective muscarinic agonist. [J] . Tecle H, Barrett SD, Lauffer DJ, Journal of Medicinal Chemistry . 1998,第14期

机译：m1-选择性毒蕈碱激动剂的设计与合成：（R）-（-）-（Z）-1-氮杂双环（2.2.1）庚烷-3-酮，O-（3-（3'-甲氧基苯基）-2-丙炔基肟肟马来酸酯（CI-1017），一种功能性m1选择性毒蕈碱激动剂。
4. One-pot conversion of azides to protected guanidines via the staudinger reduction;synthesis and utilization of the Phe-Arg hydroxyethylene dipeptide isostere [C] . Matthias Brewer, Daniel H.Rich the International Peptide Symposium . 2001

机译：通过STaudinger减少将叠氮化物转化为保护的胍; Phe-Arg羟乙烯二肽等甾醇的合成和利用
5. Part I. One-pot synthesis of secondary alcohols and one-pot asymmetric synthesis of secondary propargylic alcohols. Part II. Redox isomerization of secondary propargylic alcohols to enones. Part III. Synthesis study towards C9-C14 fragment of (+)-discodermolide. Part IV. Asymmetric synthesis of anti, anti-stereotriad building blocks for polypropionate natural products [D] . Xie, Qiuzhe 2007

机译：第一部分：仲醇的一锅法合成和仲炔丙醇的一锅法不对称合成。第二部分仲炔丙醇的氧化还原异构化为烯酮。第三部分（+）-discodermolide C9-C14片段的合成研究。第四部分聚丙烯酸酯天然产物的抗，抗立体三环构建基的不对称合成
6. Expedient one-pot synthesis of indolo32-cisoquinolines via a base-promoted N–alkylation/tandem cyclization [O] . Huy H. Nguyen, James C. Fettinger, Makhluf J. Haddadin, -1

机译：通过碱促进的N-烷基化/串联环化方便地一锅合成吲哚32-c异喹啉
7. One-Pot Eco-Safe Saccharin-Catalyzed Procedure for Expedient and Convenient Synthesis of Dihydropyrano2,3-cpyrazole, Tetrahydrobenzobpyran and Pyrano2,3-dpyrimidinone Scaffolds as a Green and Versatile Catalyst [O] . Farzaneh Mohamadpour, Mojtaba Lashkari, Nourallah Hazeri 2018

机译：用于有利和方便合成二氢吡喃的一锅生态安全糖精催化方法2,3- C 吡唑，四氢苯并 B 吡喃和吡喃2， 3- D 嘧啶酮支架作为绿色和通用催化剂

AN EXPEDIENT ONE-POT SYNTHESIS FOR PROTECTED 2-THIA-5-AZABICYCLO[2.2.1]HEPTAN-3-ONES - VERSATILE INTERMEDIATES IN THE SYNTHESIS OF CARBAPENEM SIDECHAINS

摘要

著录项

相似文献

相关主题

期刊订阅