机译:用变构结合小分子激动剂拯救人黄体生成素G蛋白偶联受体突变体的表达和信号转导
Centre for Integrative Physiology, School of Biomedical Sciences, University of Edinburgh, Edinburgh EH8 9XD, United Kingdom;
Vitrology, Glasgow G81 2LG, United Kingdom, Bristol BS1 3NY, United Kingdom;
laboratories for Integrative Neuroscience and Endocrinology (LINE), School of Clinical Sciences, University of Bristol, Bristol BS1 3NY, United Kingdom;
Department of Molecular Biophysics and Physiology, The Roy J. and Lucille A. Carver College of Medicine, University of Iowa, Iowa City, IA 52246;
Molecular Pharmacology and Drug Metabolism and Pharmacokinetics, Women's Health Department, Merck Research Laboratories, 5340 BH, Oss, The Netherlands;
Molecular Pharmacology and Drug Metabolism and Pharmacokinetics, Women's Health Department, Merck Research Laboratories, 5340 BH, Oss, The Netherlands;
Department of Molecular Biophysics and Physiology, The Roy J. and Lucille A. Carver College of Medicine, University of Iowa, Iowa City, IA 52246;
Centre for Integrative Physiology, School of Biomedical Sciences, University of Edinburgh, Edinburgh EH8 9XD, United Kingdom,University of Cape Town/Medical Research Council Group for Receptor Biology, University of Cape Town, Cape Town 7925, South Africa,Mammal Research Institute, University of Pretoria, Pretoria 0028, South Africa;
pharmacological chaperone; receptor trafficking; infertility;
机译:人黄体生成激素受体的信号选择性,纳摩尔强效变构低分子量激动剂。
机译:一种促黄体生成激素受体的信号选择性纳摩尔强效变构低分子量激动剂
机译:黄体激素受体:缓冲液成分对配体结合以及野生型和突变型受体信号传递的影响。
机译:以前 - 通过改变激动剂的信号域来拮抗G蛋白偶联肽激素受体
机译:黄体生成激素受体的同型缔合在激素介导的信号传导中的作用。
机译:用变构结合小分子激动剂拯救人黄体生成素G蛋白偶联受体突变体的表达和信号转导
机译:用变构结合小分子激动剂拯救人黄体生成素G蛋白偶联受体突变体的表达和信号转导