机译:新型大脑调节剂将GSPT1募集到CRL4(CRBN)泛素连接酶
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Tokyo Med Univ, Dept Nanoparticle Translat Res, Shinjuku Ku, Tokyo 1608402, Japan;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Scripps Res Inst, San Diego, CA 92121 USA;
Scripps Res Inst, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Tokyo Med Univ, Dept Nanoparticle Translat Res, Shinjuku Ku, Tokyo 1608402, Japan;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
Celgene Corp, 10300 Campus Point Dr,Suite 100, San Diego, CA 92121 USA;
机译:蛋白质降解通过CRL4 CRBN sup>泛素连接酶:促进AIOLOS和/或GSPT1的降解的新型戊二胺类似物的发现和结构 - 活性关系
机译:CRL4(CRBN)泛素连接酶对来那度胺诱导的CK1α降解的结构基础
机译:DDB1-CRBN E3泛素连接酶与沙利度胺复合的结构:洞察小分子对CRL4的抑制作用
机译:鉴定参与乳腺癌发病的E3泛素连接酶的靶类似物:一种合理的药物设计方法
机译:泛素连接酶Hrd1p与泛素结合酶Ubc7p的功能分析。
机译:c-Abl激酶的激活通过促进DDA1蛋白募集到CRL4泛素连接酶来增强抗骨髓瘤药物来那度胺的活性。
机译:教师观点通过调节E3泛素连接酶复合CRL4(CRBN)来诱导T细胞阻遏物Ikaros和AIOLOS的降解来推荐免疫调节剂和吡喃胺和吡啶胺共刺激T细胞的推荐。