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Innovative Tilidine-Naloxone Sustained Release Drug Delivery Systems based on Kollicoat? Polymers

机译:基于Kollicoat的创新的Tilidine-Naloxone缓释药物递送系统?聚合物

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Tilidine/naloxone single unit drug delivery systems were developed by coating of directly compressed immediate release cores with an extremely flexible combination of Kollicoat? SR 30 D and Kollicoat? IR. The Kollicoat? DDS formulations released both actives simultaneously and more constantly than marketed products. Drug release can be adjusted in wide ranges mainly by altering the ratio of lipophilic to hydrophilic polymer and the coating level.
机译:通过直接压缩的立即释放核心和极其灵活的Kollicoid组合,开发了Tilidine / Naloxone单位药物递送系统? SR 30 D和Kollicoat? IR。 Kollicoat? DDS制剂同时释放了两个活性,而不是市场产品。可以主要通过改变亲水性聚合物和涂层水平的亲脂性比例来调节药物释放。

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