首页> 外国专利> R-3-3S4S-3--4-4--1--1-4--2- R-3-3S4S-3-FLUORO-4-4-HYDROXYPHENYLPIPERIDIN-1-YL-1-4-METHYLBENZYLPYRROLIDIN-2-ONE AND ITS PRODRUGS FOR THE TREATMENT OF PSYCHIATRIC DISORDERS

R-3-3S4S-3--4-4--1--1-4--2- R-3-3S4S-3-FLUORO-4-4-HYDROXYPHENYLPIPERIDIN-1-YL-1-4-METHYLBENZYLPYRROLIDIN-2-ONE AND ITS PRODRUGS FOR THE TREATMENT OF PSYCHIATRIC DISORDERS

机译:r-3-3s4s-3--4-4--1--1-4--2-r-3-3s4s-3-fluoro-4-4-羟基苯基哌啶-1-基1-4-甲基苄基吡咯烷 - 2- one及其前药治疗精神病疾病

摘要

The present disclosure relates generally to compounds of formula (I), including salts thereof, and to compositions and methods of using such compounds. The compounds are ligands of the NR2B NMDA receptor and may be useful in the treatment of various central nervous system disorders.
机译:本公开一般涉及式(I)化合物,包括其盐,以及使用这些化合物的组合物和方法。 该化合物是NR2B NMDA受体的配体,可用于治疗各种中枢神经系统障碍。

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