首页> 外国专利> SOLID FORMS OF 3-((1R,3R)-1-(2,6-DIFLUORO-4-((1-(3-FLUOROPROPYL)AZETIDIN-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO3,4-BINDOL-2-YL)-2,2-DIFLUOROPROPAN-1-OL AND PROCESSES FOR PREPARING FUSED TRICYCLIC COMPOUNDS COMPRISING A SUBSTITUTED PHENYL OR PYRIDINYL MOIETY, INCLUDING METHODS OF THEIR USE

SOLID FORMS OF 3-((1R,3R)-1-(2,6-DIFLUORO-4-((1-(3-FLUOROPROPYL)AZETIDIN-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO3,4-BINDOL-2-YL)-2,2-DIFLUOROPROPAN-1-OL AND PROCESSES FOR PREPARING FUSED TRICYCLIC COMPOUNDS COMPRISING A SUBSTITUTED PHENYL OR PYRIDINYL MOIETY, INCLUDING METHODS OF THEIR USE

机译:3 - ((1R,3R)-1-(2,6-二氟-4-((1-(3-氟丙基)氮杂萘-3-基)氨基)苯基)-3-甲基-1,3 ,4,9-四氢-2H-吡啶[3,4-B]吲哚-2-基)-2,2-二氟丙烷-1-醇和制备包含取代苯基或吡啶基部分的熔融三环化合物的方法,包括方法他们的使用

摘要

Provided herein are solid forms, salts such as compound B, and formulations of 3-((lR,3R)-l-(2,6-difluoro-4-((l-(3-fluoropropyl) azetidin-3-yl)amino)phenyl)-3-methyl-l,3,4,9-tetrahydro-2H- pyrido[3,4-b]indol-2-yl)-2,2-difluoropropan-l-ol, processes and synthesis thereof, and methods of their use in the treatment of cancer.
机译:本文提供了固体形式,盐,如化合物B,以及3 - ((LR,3R)-1-(2,6-二氟-4-((L-(3-氟丙基)氮素-3-y1)氨基)苯基)-3-甲基-1,3,4,9-四氢-2H-吡啶[3,4-B]吲哚-2-基)-2,2-二氟丙烷-1-醇,方法和合成以及它们在治疗癌症时使用的方法。

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