embedded image ;can be used to make antibody-drug conjugates. The conjugates so made are stable in both human and mouse serum, enabling the performance of pre-clinical studies using a mouse model."/> MODIFIED SELF-IMMOLATING MOIETIES FOR USE IN PRODRUGS AND CONJUGATES AND METHODS OF USING AND MAKING
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MODIFIED SELF-IMMOLATING MOIETIES FOR USE IN PRODRUGS AND CONJUGATES AND METHODS OF USING AND MAKING

机译:改性自焚部分用于前药和共轭和使用和制造方法

摘要

Compounds represented by formula (I); embedded image ;can be used to make antibody-drug conjugates. The conjugates so made are stable in both human and mouse serum, enabling the performance of pre-clinical studies using a mouse model.
机译:由式(I)表示的化合物; <化学ID =“Chem-US-00001”> “嵌入式图像”文件=“US20210113706A1-20210422-C00001.gif”他=“30.73mm”ImgContent ;可用于制备抗体 - 药物缀合物。如此制备的缀合物在人和小鼠血清中稳定,可以使用小鼠模型进行临床前研究的性能。

著录项

  • 公开/公告号US2021113706A1

    专利类型

  • 公开/公告日2021-04-22

    原文格式PDF

  • 申请/专利权人 BRISTOL-MYERS SQUIBB COMPANY;

    申请/专利号US202017126555

  • 发明设计人 YAM B. POUDEL;SANJEEV GANGWAR;

    申请日2020-12-18

  • 分类号A61K47/65;A61K47/64;A61K47/68;A61P35;A61K45/06;

  • 国家 US

  • 入库时间 2022-08-24 18:20:31

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