首页> 外国专利> USE OF EZH2 INHIBITOR COMBINED WITH CDK4/6 INHIBITOR IN PREPARATION OF DRUG FOR TREATING TUMOR

USE OF EZH2 INHIBITOR COMBINED WITH CDK4/6 INHIBITOR IN PREPARATION OF DRUG FOR TREATING TUMOR

机译:EZH2抑制剂联合CDK4 / 6抑制剂在制备药物治疗肿瘤中的用途

摘要

The present invention relates to use of an EZH2 inhibitor combined with a CDK4/6 inhibitor in the preparation of a drug for treating a tumor. Specifically, the EZH2 inhibitor involved in the present invention is selected from a compound shown in formula (I) or a pharmaceutically acceptable salt thereof, and the involved CDK4/6 inhibitor is selected from a compound shown in formula (II) or a pharmaceutically acceptable salt thereof. Compared with a single drug, the combination of the EZH2 inhibitor and the CDK4/6 inhibitor further enhances the anti-tumor effect.
机译:本发明涉及EZH2抑制剂与CDK4 / 6抑制剂联合的用途在制备用于治疗肿瘤的药物中。具体地,本发明中涉及的EZH2抑制剂选自式(I)中所示的化合物,或其药学上可接受的盐,并且所涉及的CDK4 / 6抑制剂选自式(II)中所示的化合物或药学上可接受的化合物盐。与单一药物相比,EZH2抑制剂和CDK4 / 6抑制剂的组合进一步增强了抗肿瘤作用。

著录项

  • 公开/公告号WO2021063332A1

    专利类型

  • 公开/公告日2021-04-08

    原文格式PDF

  • 申请/专利权人 JIANGSU HENGRUI MEDICINE CO. LTD.;

    申请/专利号WO2020CN118612

  • 发明设计人 ZHANG LAN;LIAO CHENG;

    申请日2020-09-29

  • 分类号A61K31/4545;A61K31/4433;A61K31/519;C07D405/14;C07D471/04;A61P35;

  • 国家 CN

  • 入库时间 2022-08-24 18:09:54

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