首页> 外国专利> INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS

INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS

机译：吲哚羧酰胺衍生物作为P2X7受体拮抗剂

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摘要

The present invention relates to indole carboxamide derivatives of formula (I), their preparation and their use as pharmaceutically active compounds: [In the formula, R¹ , R² , R³ , R⁴ , R⁵ and R⁶ are as defined in the specification].

机译：本发明涉及式（I）的吲哚羧胺衍生物，其制备及其作为药物活性化合物的用途：[在式中， R + 1 ， r 2 ， r 3 ， r 4 ， R 5 和< b> r 6 在规范中定义]。 展开▼

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公开/公告号KR102232742B1

专利类型

公开/公告日2021-03-26

原文格式PDF

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申请/专利号KR1020157018405

发明设计人 힐퍼트 쿠르트;위블레 프랑시스;깽메를랭 티에리;렌네베르크 도르테;슈탐 지몬;
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申请日2013-12-11

分类号C07D209/08;A61K31/404;A61K31/4155;A61K31/422;A61K31/506;C07D403/12;C07D403/14;C07D413/12;C07D413/14;C07D417/12;C07D498/08;

国家 KR

入库时间 2022-08-24 17:57:25

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1. 作为P2X7受体拮抗剂的吲哚羧酰胺衍生物 [P] . 中国专利： CN104812749B . 2016.12.14

2. 作为P2X7受体拮抗剂的吲哚羧酰胺衍生物 [P] . 中国专利： CN104812749A . 2015-07-29

3. INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS [P] . KR102232744B1 . 2021-03-26

机译：吲哚羧酰胺衍生物作为P2X7受体拮抗剂

4. INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS [P] . CA2890886C . 2020-10-27

机译：吲哚羧酰胺衍生物作为P2X7受体拮抗剂

5. INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS. [P] . MX368044B . 2019-09-17

机译：吲哚羧酰胺衍生物作为P2X7受体拮抗剂。

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