首页> 外国专利> C-NUCLEOSIDES, C-NUCLEOTIDES AND THEIR ANALOGS, EQUIVALENTS AND PRODRUGS THEREOF FOR ECTONUCLEOTIDASE INHIBITION

C-NUCLEOSIDES, C-NUCLEOTIDES AND THEIR ANALOGS, EQUIVALENTS AND PRODRUGS THEREOF FOR ECTONUCLEOTIDASE INHIBITION

机译:C-核苷,C-核苷酸及其类似物,其等当量和前药,用于异构核苷酸酶抑制

摘要

The invention provides novel heterocyclic C-nucleosides, C-nucleotides and their analogues, equivalents, and prodrug thereof. The compounds, compositions, and methods provided of the invention, by themselves or in combination with other therapies are useful for the treatment of a disease, disorder or condition related to CD73 (ecto-5'-nucleotidase) enzyme.
机译:本发明提供了新型杂环C-核苷,C核苷酸及其类似物,等同物和前药。本发明提供的本发明或与其他疗法组合的化合物,组合物和方法可用于治疗与CD73(ECTO-5'-核苷酸酶)酶相关的疾病,病症或病症。

著录项

  • 公开/公告号WO2021040356A1

    专利类型

  • 公开/公告日2021-03-04

    原文格式PDF

  • 申请/专利权人 KAINOS MEDICINE INC.;

    申请/专利号WO2020KR11268

  • 申请日2020-08-24

  • 分类号C07H21/02;A61K31/7076;A61K31/706;A61P35;

  • 国家 KR

  • 入库时间 2022-08-24 17:32:24

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