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Therapeutic agent and compositions having the inhibitory action for ª‰-glucuronidase and method of inhibiting ª‰-glucuronidase

机译:对β-葡糖醛酸糖苷酶具有抑制作用的治疗剂和组合物以及抑制β-葡糖醛酸糖苷酶的方法

摘要

Pharmaceutical compositions having b -glucuronidase-inhibiting activity comprise a carrier and 2,5-di-O-acetyl D-glucosaccharo-1,4-3,6-dilactone. They may be in forms suitable for oral, parenteral or rectal administration and may comprise a b -group vitamin or vitamin C or a glucuronic acid derivative e.g. p D-glucuronolactone or D-glucuronamide in addition to conventional diluents and excipients.
机译:具有β-葡糖醛酸糖苷酶抑制活性的药物组合物包含载体和2,5-二-O-乙酰基D-葡萄糖基-1,4-3,6-二内酯。它们可以是适合口服,肠胃外或直肠给药的形式,并且可以包含b族维生素或维生素C或葡糖醛酸衍生物,例如维生素B。除常规稀释剂和赋形剂外,p D-葡萄糖醛酸内酯或D-葡萄糖醛酸酰胺。

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