Psycholeptic benzodiazepines.. M3A. Are new compounds of formula: (R', R2, R3 = H, alkyl, alkoxy, halogen, OH, NO2, CN, acyl, CF3, NH2, acylamino, alkylamino, dialkylamino, acyloxy, COOH, alkoxycarbonyl, CONH2, CONH.alkyl, CON(alkylthio, alkylsulphinyl, alkylsulphonyl; R4 = H, alkyl, cycloalkyl, aralkyl, aryl, phenacyl; R5 = H, alkyl; A = alkylene; Y = O or S). Used as tranquillisers, sedatives and anti-depressants. Low toxicity with few side effects in man. The are prepared as follows:-.
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机译：精神安定的苯二氮卓类药物.. M3A。是下式的新化合物：（R'，R2，R3 = H，烷基，烷氧基，卤素，OH，NO2，CN，酰基，CF3，NH2，酰基氨基，烷基氨基，二烷基氨基，酰氧基，COOH，烷氧羰基，CONH2，CONH。烷基，CON（烷硫基，烷基亚磺酰基，烷基磺酰基; R4 = H，烷基，环烷基，芳烷基，芳基，苯甲酰基; R5 = H，烷基; A =亚烷基; Y = O或S）。用作镇定剂，镇静剂和抗抑郁药。低毒，对人体几乎没有副作用。
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