2-Amino-1,5-benzodiazocines and 5-oxides thereof - having CNS active props

摘要

Benzodiazocines have general formula (I): (R1 = H, halo, CF3, CN, NO2, or 1-6C alkoxy, alkyl or alkylthio, R2 = H, 1-6C alkyl, or furyl, R3 = H, 1-6C alkyl, 1-6C hydroxyalkyl, 2-6C alkenyl, or benzyl, A = R4 = phenyl, (1-6C alkyl)-phenyl, nitrophenyl, halophenyl or pyridyl) and they are their salts are tranquillizers, sedatives, anticonvulsants, and hypnotics as well as possible diuretics and anti-inflammatories.