2.9 - dioxatricyclo (4,3,1,0,3,7) deans and method for preparation thereof.

摘要

4-amino-3-methyl-2,9-dioxatricyclo[4,3,1,03,7]decane derivatives are disclosed which exhibit analgesic properties, and which have the formula (I) IMAGE (I) wherein ONE OF R1 and R2 represents hydrogen and the other represents an amino group which is substituted by an arylalkyl group or an arylalkenyl group, ONE OF R3 and R4 represents hydrogen and the other represents alkoxy, and Y AND Y' EACH REPRESENT HYDROGEN OR JOINTLY FORM A BOND, AND PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF, AS WELL AS PHARMACEUTICAL FORMULATIONS THEREOF.