首页> 外国专利> NB QUARTERLY DERIVATIVES OF 10-BROMAJMALINE AND 10-BROMISOAJMALINE SOFT PROCEDURE AND INTERMEDIATES FOR THE PREPARATION OF THESE DERIVATIVES

NB QUARTERLY DERIVATIVES OF 10-BROMAJMALINE AND 10-BROMISOAJMALINE SOFT PROCEDURE AND INTERMEDIATES FOR THE PREPARATION OF THESE DERIVATIVES

机译:NB 10-溴香豆碱和10-溴香豆碱软方法的季衍生物和中间体,用于制备这些衍生物

摘要

New quaternary derivatives of 10-bromoajmaline and 10-bromoisoajmaline are disclosed which exhibit antiarrhythmic and adrenolytic properties and which have the formula I IMAGE (I) wherein R represents a carbon-attached organic group containing 1 to 10 carbon atoms and A- represents an acid anion as well as pharmaceutical formulations thereof and processes and intermediates for their preparation.
机译:公开了具有抗心律不齐和肾上腺素解性质的10-溴代间苯二胺和10-溴代异间苯二胺的新季衍生物,其具有式I (I),其中R代表含碳原子的有机基团,含1至10个碳原子,A-代表酸阴离子及其药物制剂及其制备方法和中间体。

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