首页> 外国专利> PROCESS FOR THE PREPARATION OF NEW BENZOYLUREA COMPOUNDS AND OF COMPOSITIONS CONTAINING SAME BEING SOME OF THEM ACTIVE IN THE CONTROL OF MITES WHITEFLY AND THRIPS AND OTHERS PHARMACEUTICAL ONES DESTINED TO COMBAT TUMORS IN LIVING BEINGS AS WELL AS FOR THE UTILIZATION OF SAME

PROCESS FOR THE PREPARATION OF NEW BENZOYLUREA COMPOUNDS AND OF COMPOSITIONS CONTAINING SAME BEING SOME OF THEM ACTIVE IN THE CONTROL OF MITES WHITEFLY AND THRIPS AND OTHERS PHARMACEUTICAL ONES DESTINED TO COMBAT TUMORS IN LIVING BEINGS AS WELL AS FOR THE UTILIZATION OF SAME

机译:制备新的苯甲脲类化合物及其组成的方法,其中一些活性成分可有效控制矿山和节律以及其他与矿物质有竞争性的矿物质,同时也用于其用途

摘要

The invention relates to a composition active against mites, whitefly and thrips, which comprises, in addition to a liquid or solid inert carrier material, a benzoylurea compound of the general formula IMAGE wherein R1 is hydrogen atom or represents 1 or 2 substituents which are selected from the group consisting of chlorine, methyl and trifluoromethyl, R2 is an alkyl group having 2-4 carbon atoms or a cycloalkyl group having 3 or 4 carbon atoms, R3 is a hydrogen atom or represents 1-3 substituents which are selected from the group consisting of halogen, and alkyl, alkoxy, haloalkyl and haloalkoxy having 1-4 carbon atoms, R4 and R5 are both fluorine atoms, or wherein R4 is a chlorine atom and R5 is a hydrogen atom, and X is an oxygen or sulphur atom. The composition may be used in a dosage of 10 to 5000 g of active substance per hectare. The invention further relates to pharmaceutical compositions comprising the above compounds. Finally the invention relates to new benzoylurea compounds and to the preparation thereof.
机译:本发明涉及对螨,粉虱和蓟马有活性的组合物,该组合物除了液体或固体惰性载体材料外,还包含通式为的苯甲酰脲化合物,其中R1为氢原子或代表1或2个取代基,选自氯,甲基和三氟甲基,R 2是具有2-4个碳原子的烷基或具有3或4个碳原子的环烷基,R 3是氢原子或代表1-3个选自以下的取代基卤素和具有1-4个碳原子的烷基,烷氧基,卤代烷基和卤代烷氧基组成的基团,R4和R5均为氟原子,或其中R4为氯原子且R5为氢原子,且X为氧或硫原子。所述组合物可以每公顷10至5000g活性物质的剂量使用。本发明进一步涉及包含上述化合物的药物组合物。最后,本发明涉及新的苯甲酰脲化合物及其制备。

著录项

  • 公开/公告号PT77990A

    专利类型

  • 公开/公告日1984-02-01

    原文格式PDF

  • 申请/专利权人 DUPHAR INTERNATIONAL RESEARCH B.V.;

    申请/专利号PT19840077990

  • 发明设计人

    申请日1984-01-20

  • 分类号C07C;A01N;A61K;

  • 国家 PT

  • 入库时间 2022-08-22 09:13:55

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号