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BENZOYLUREA COMPOUNDS, COMPOSITION HAVING INSECTICIDE AND ACARICIDE ACTIVITY, PHARMACEUTICAL COMPOSITION, PROCESS TO CONTROL INSECTS AND / OR MITES AND PROCESS TO COMBAT TUMORS IN LIVING BEINGS
BENZOYLUREA COMPOUNDS, COMPOSITION HAVING INSECTICIDE AND ACARICIDE ACTIVITY, PHARMACEUTICAL COMPOSITION, PROCESS TO CONTROL INSECTS AND / OR MITES AND PROCESS TO COMBAT TUMORS IN LIVING BEINGS
The invention relates to new benzoylurea compounds of the general formula IMAGE wherein R1 is a halogen atom, R2 is a hydrogen atom or a halogen atom, R3 is a hydrogen atom or represents 1 or 2 substituents which are selected from the group consisting of chlorine, methyl and trifluoromethyl, R4 is a hydrogen atom, an alkyl group having 1-6 carbon atoms or a cycloalkyl group having 3-6 carbon atoms, R5 is a hydrogen atom or an alkyl group having 1-4 carbon atoms, and A is a phenyl group or a heteroaryl group having 1 or 2 nitrogen atoms, which groups may be substituted with 1-3 substituents which are selected from the group consisting of halogen, and alkyl, alkoxy, haloalkyl and haloalkoxy having 1-4 carbon atoms. The compounds have an insecticidal and acaricidal activity. After having been processed to compositions, the compounds may be used for control of insects and/or mites in a dosage from 1 to 5000 g of active substance per hectare. In addition the compounds have an anti-tumor activity and may be used in pharmaceutical compositions.
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机译:本发明涉及通式的新的苯甲酰脲化合物,其中R 1是卤素原子,R 2是氢原子或卤素原子,R 3是氢原子或代表1或2个选自以下的取代基:氯,甲基和三氟甲基,R4为氢原子,碳数为1-6的烷基或碳原子数为3-6的环烷基,R5为氢原子或碳数为1-4的烷基,A R 1为具有1或2个氮原子的苯基或杂芳基,其基团可被1-3个取代基取代,所述取代基选自卤素,以及具有1-4个碳原子的烷基,烷氧基,卤代烷基和卤代烷氧基。该化合物具有杀虫和杀螨活性。在加工成组合物之后,该化合物可以以每公顷1至5000g活性物质的剂量用于防治昆虫和/或螨。另外,该化合物具有抗肿瘤活性,可以用于药物组合物中。
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