首页> 外国专利> MORPHOLINYL DERNORUBICIN DERIVATIVES, MORPHOLINYL DOXORUBICIN DERIVATIVES AND THEIR ANALOGS AND THEIR ANTITUMOR APPLICATION

MORPHOLINYL DERNORUBICIN DERIVATIVES, MORPHOLINYL DOXORUBICIN DERIVATIVES AND THEIR ANALOGS AND THEIR ANTITUMOR APPLICATION

机译:吗啉基去污柔比星衍生物,吗啉基阿霉素变质及其类似物和其抗肿瘤应用

摘要

The present invention has as its object new industrial compounds. These compounds have the following structure: BR/ BR/ BR/ BR BR BR BR BR R IS CHOSEN IN THE GROUP CONSISTING OF -CO-CH, -CHOH-CH, -CO-CHOH, -CHOH-CHOH, ETC., HYDROGEN OR METHOXY; / P P XO OR NH; / P P R AND R TOGETHER H, OH OR METHOXY; / P P A IS A HYDROGEN OR A CYANO; / P P ZO, S, ETC / P p THESE DERIVATIVES HAVE ANTITUMOR APPLICATION.
机译:本发明的目的是新型工业化合物。这些化合物具有以下结构:







在由-CO-CH,-CHOH-组成的基团中R被选择CH,-CO-CHOH,-CHOH-CHOH等,氢或甲氧基; P> XO或NH;

R和R一起为H,OH或甲氧基;

A是氢或氰基;

ZO,S,ETC >这些衍生物具有反面的应用。

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