首页> 外国专利> PEPTIDES AND PEPTIDE DERIVATIVES, THEIR PREPARATION, THEIR USE IN THERAPEUTICS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

PEPTIDES AND PEPTIDE DERIVATIVES, THEIR PREPARATION, THEIR USE IN THERAPEUTICS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

机译:肽和肽衍生物,其制备,在包含相同成分的治疗药物和药物组合物中的使用

摘要

P THE INVENTION CONCERNS PEPTIDES POSSIBLY IN THE ISOSTERATED FORM IN WHICH A METHYLENE GROUP LOCATED IN THE CHAIN IS DISUBSTITUTED, ONE OF THE SUBSTITUENTS OR BOTH OF WHICH IS FLUORINE AND CHLORINE. / P P THESE COMPOUNDS MAY BE USED AS MEDICINES, ESPECIALLY AS INHIBITORS OF THE RENINE. / P
机译:

本发明以肽形式存在于肽中,该肽以位于链中的亚甲基被取代,氟和氯的一种或两种取代物取代。

这些化合物可以用作药物,尤其是作为肾素的抑制剂。

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