首页> 外国专利> 6(R)-(2-(8'-ACYLOXY-2'-METHYL-6'-METHYL(OR HYDROGEN)-POLYHYDRONAPHTHYL-1')-ETHYL)-4(R)-HYDROXY-3,4,5,6-TETRAHYDRO-2H-PYRAN-2-ONES,THE HYDROXY ACID FORM OF SAID PYRANONES,THE PHARMACEUTICALLY ACCEPTABLE SALTS OF SAID HYDROXY ACIDS,AND THE LOWER ALKYL,AND PHENYL,DIMETHYLAMINO OR ACETYLAMINO SUBSTITUTED LOWER ALKYL ESTERS OF SAID HYDROXY ACID,PROCESSES FOR PREPARING THE SAME, AND A PHARMACEUTICAL ANTIHYPERCHOLESTEROLEMIC COMPOSITION CONTAINING THE SAME

6(R)-(2-(8'-ACYLOXY-2'-METHYL-6'-METHYL(OR HYDROGEN)-POLYHYDRONAPHTHYL-1')-ETHYL)-4(R)-HYDROXY-3,4,5,6-TETRAHYDRO-2H-PYRAN-2-ONES,THE HYDROXY ACID FORM OF SAID PYRANONES,THE PHARMACEUTICALLY ACCEPTABLE SALTS OF SAID HYDROXY ACIDS,AND THE LOWER ALKYL,AND PHENYL,DIMETHYLAMINO OR ACETYLAMINO SUBSTITUTED LOWER ALKYL ESTERS OF SAID HYDROXY ACID,PROCESSES FOR PREPARING THE SAME, AND A PHARMACEUTICAL ANTIHYPERCHOLESTEROLEMIC COMPOSITION CONTAINING THE SAME

机译:6(R)-(2-(8'-酰基-2'-甲基-6'-甲基(或氢)-聚乙烯基萘-1')-乙基)-4(R)-羟基-3,4,5, 6-四氢-2H-吡喃-2-酮,硬脂酸吡喃酮的羟基形式,硬脂酸的药学上可接受的盐,低级烷基和被取代的苯甲基,二甲基酰胺基或乙酰氨基缩水甘油用于制备相同的药物,以及包含相同的药物的抗胆甾醇成分

摘要

机译:

著录项

  • 公开/公告号KE3746A

    专利类型

  • 公开/公告日1987-10-02

    原文格式PDF

  • 申请/专利权人 MERCK & CO. INC.;

    申请/专利号KE19870003746

  • 申请日1987-08-14

  • 分类号C07D309/30;A61K31/22;A61K31/365;C07C59/11;C07C69/30;

  • 国家 KE

  • 入库时间 2022-08-22 07:20:10

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