首页> 外国专利> VASCULOPROTECTIVE PHARMACEUTICAL COMPOSITIONS CONTAINING A UBIQUINONE DERIVATIVE AND AT LEAST ONE OTHER COMPOUND HAVING A VASCULOPROTECTIVE ACTIVITY

VASCULOPROTECTIVE PHARMACEUTICAL COMPOSITIONS CONTAINING A UBIQUINONE DERIVATIVE AND AT LEAST ONE OTHER COMPOUND HAVING A VASCULOPROTECTIVE ACTIVITY

机译:包含泛醌衍生物和至少一种具有血管保护活性的其他化合物的血管保护药物组合物

摘要

PHARMACEUTICAL COMPOSITIONS HAVING VASCULOPROTECTIVE ACTIVITY CONTAINING A UBIQUINONE DERIVATIVE AND AT LEAST ONE OTHER COMPOUND HAVING KNOWN VASCULOPROTECTIVE ACTIVITY. PREFERABLY, THE UBIQUINONE DERIVATIVE IS COENZYME Q. / P P ADVANTAGEALLY, KNOWN COMPOUNDS HAVING VASCULOPROTECTIVE ACTIVITY ARE CHOSEN AMONG COMPOUNDS HAVING FLAVONOID, HEPARINOID, TERPENIC OR GLUCOSIDIC STRUCTURE, AND MORE PREFERABLY, IN THE GROUP COMPRISING: RUTIN, O- (B-HYDROXYETHYLRUTOSIDE), DELPHINIDINE, HESPERIDINE, DIOSMINE, ASIATICOSIDE, CATECHIN, HEPARIN, ESCIN, RUSCOGENINE, TRIBENOSIDE, SODIUM 2-PHENYL-5,7-DIOXYACETATE, BENZO-G-PYRONE. / P P COENZYME Q AND VASCULOPROTECTIVE COMPOUND MAY BE PRESENT IN REPORTS VARYING FROM 1: 1 TO 1: 1000. COMPOSITIONS ACCORDING TO THE INVENTION MAY BE ADMINISTERED ORAL, PARENTERAL, RECTAL OR TOPICAL, IN THE FORM OF CAPSULES, TABLETS, SYRUPS, PELLETS, STERILE SOLUTIONS, OINTMENTS, CREAMS, LOTIONS, GELS OR SUPPOSITORIES. / P OBSERVED, UNEXPECTEDLY, A SYNERGY OF THE THERAPEUTIC EFFECTS OF COMPONENTS WITHOUT AGGRAVATING THE TOXICITY.
机译:具有包含泛泛酮衍生物的血管保护活性且至少一种具有已知的血管保护活性的其他化合物的药物组合物。泛醌衍生物最好是辅酶Q。 (B-羟基乙氧基核糖苷),苯乙胺啶,橙皮碱,薯OS碱,阿糖胺苷,儿茶素,肝素,毛细血管生成素,松香碱,三苯乙内酯,2-苯基-5,7-二氧己酸酯钠,苯并-G-吡啶酮。

辅酶Q和血管保护性化合物的比例可能为1:1至1:1000。根据本发明的成分可能以胶囊,片剂的形式口服,口服,直肠,直肠或局部给药,糖浆,丸剂,无菌溶液,药膏,乳霜,乳液,乳液或栓剂。 意外地观察到了在不吸收毒性的情况下对组件的治疗效果的协同作用。

著录项

  • 公开/公告号FR2587212A1

    专利类型

  • 公开/公告日1987-03-20

    原文格式PDF

  • 申请/专利权人 SEUREF AG;SEUREF AG;

    申请/专利号FR19860006270

  • 发明设计人 BRASEY PIERRE-NOEL;PIERRE-NOEL BRASEY;

    申请日1986-04-30

  • 分类号A61K31/12;A61K31/70;A61K31/725;A61K45/06;

  • 国家 FR

  • 入库时间 2022-08-22 07:11:15

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