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SYNTHESIS OF INOTROPIC IMIDAZOÛ4,5-C¨PYRIDINE
SYNTHESIS OF INOTROPIC IMIDAZOÛ4,5-C¨PYRIDINE
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机译:内生咪唑Û4,5-吡啶的合成
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摘要
The present invention provides a process for preparing 2-[2-methoxy-4-(methylthio)phenyl]-1(3)H-imidazo[4,5-c]pyridine comprising reacting 3,4-diaminopyridine with 2-methoxy-4-methylthiobenzoic acid in the presence of phosphorus oxychloride and pyridine.
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