首页> 外国专利> 8, 9-FUSED DHYDRO-BETA-CARBORIC ACID DERIVATIVE, 8, 9-FUSED 3, 4-BETA-CARBORIC ACID DERIVATIVE, PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF, PHARMACEUTICAL COMPOSITION, CLOT DISSOLVING OR PREVENTING METHOD AND PRODUCTION OF CARBORIC ACID DERIVATIVE

8, 9-FUSED DHYDRO-BETA-CARBORIC ACID DERIVATIVE, 8, 9-FUSED 3, 4-BETA-CARBORIC ACID DERIVATIVE, PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF, PHARMACEUTICAL COMPOSITION, CLOT DISSOLVING OR PREVENTING METHOD AND PRODUCTION OF CARBORIC ACID DERIVATIVE

机译:8,8,9-氟-BETA羧酸衍生物,8,9-氟3,4-BETA羧酸衍生物,药理学上可接受的盐,药物成分,溶解或防止污渍的方法和生产方法

摘要

The invention relates to a group of new 8,9-annelated- beta -carbolines and 8,9-annelated-3,4-dihydro- beta -carbolines having interesting fibrinolytic properties. In particular the compounds can be used as orally active fibrinolytics. The compounds have the general formulae 1 and 2 CHEM wherein R2 + R3 together with the carbon atom and the nitrogen atom to which they are bound and the intermediate carbon atom constitute a heterocyclic group consisting of 5-10 ring atoms.
机译:本发明涉及一组新的具有有趣的纤溶特性的8,9-退火的β-咔啉和8,9-退火的3,4-二氢-β-咔啉。特别地,所述化合物可用作口服活性纤溶剂。所述化合物具有通式1和2 ,其中R 2 + R 3与它们所键合的碳原子和氮原子以及中间碳原子一起构成由5-10个环原子组成的杂环基。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号