wherein R¹ is hydrogen, (C₁-C₅) alkyl, (C₁-C₃) haloalkyl or halogen; R², R³ independently of each other (C₁-C₅) alkyl, (C₂-C₅) alkenyl, (C₂-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) - haloalkyl, halogen, cyano, nitro, (C₁-C₅) alkoxy, (C₁-C₃) alkoxy (C₁-C₃) alkyl, (C₁-C₃) -haloalkoxy, (C₁-C₃) alkylthio, or R² and R³ together form a polymethylene chain of 2 to 5 carbon atoms; R⁴ is hydrogen, (C₁-C₁₀) alkyl, (C₂-C₅) alkenyl, (C₃-C₇) -cycloalkyl; R⁵ is hydrogen, (C₁-C₁₀) alkyl, (C₃-C₅) alkenyl, (C₃-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) -haloalkyl or (C₁-C₃) alkoxy (C₁-C₃) alkyl, X is oxygen, sulfur or a -NR⁶ group; R⁶ is hydrogen, (C₁-C₅) alkyl, (C₃-C₅) alkenyl, (C₃-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) -haloalkyl or (C₁-C₃) alkoxy (C₁-C₃) alkyl mean and include their biologically acceptable acid addition salts.; The compounds of formula I are novel and are also encompassed by the invention."/> Agents containing imidazoline derivatives for the control, based on the host animal system, of ectoparasites, and these imidazolines derivatives
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Agents containing imidazoline derivatives for the control, based on the host animal system, of ectoparasites, and these imidazolines derivatives

机译:包含咪唑啉衍生物的药物,用于根据宿主动物系统控制外寄生虫和这些咪唑啉衍生物

摘要

The present invention is intended to wirtstiersystemischen controlling ectoparasites, characterized in that it comprises a compound of formula I wherein R¹ is hydrogen, (C₁-C₅) alkyl, (C₁-C₃) haloalkyl or halogen; R², R³ independently of each other (C₁-C₅) alkyl, (C₂-C₅) alkenyl, (C₂-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) - haloalkyl, halogen, cyano, nitro, (C₁-C₅) alkoxy, (C₁-C₃) alkoxy (C₁-C₃) alkyl, (C₁-C₃) -haloalkoxy, (C₁-C₃) alkylthio, or R² and R³ together form a polymethylene chain of 2 to 5 carbon atoms; R⁴ is hydrogen, (C₁-C₁₀) alkyl, (C₂-C₅) alkenyl, (C₃-C₇) -cycloalkyl; R⁵ is hydrogen, (C₁-C₁₀) alkyl, (C₃-C₅) alkenyl, (C₃-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) -haloalkyl or (C₁-C₃) alkoxy (C₁-C₃) alkyl, X is oxygen, sulfur or a -NR⁶ group; R⁶ is hydrogen, (C₁-C₅) alkyl, (C₃-C₅) alkenyl, (C₃-C₅) alkynyl, (C₃-C₇) -cycloalkyl, (C₃-C₇) cycloalkenyl, (C₁-C₃) -haloalkyl or (C₁-C₃) alkoxy (C₁-C₃) alkyl mean and include their biologically acceptable acid addition salts.; The compounds of formula I are novel and are also encompassed by the invention.
机译:本发明意在使系统控制外寄生虫,其特征在于它包括式Ⅰ化合物:其中R 1是氢,(C 1 -C 4)烷基,(C 1 -C 4)卤代烷基或卤素; R 2,R 3彼此独立(C 1 -C 4)烷基,(C 2 -C 4)烯基,(C 2 -C 4)炔基,(C 1 -C 4)-环烷基,(C 1 -C 4)环烯基,(C 1 -C 4)-卤代烷基,卤素,氰基,硝基,(C 1 -C 4)烷氧基,(C 1 -C 4)烷氧基(C 1 -C 4)烷基,(C 1 -C 4)-卤代烷氧基,(C 1 -C 4)烷硫基或R 2和R 3一起形成聚亚甲基2至5个碳原子的链; R 5是氢,(C 1 -C 4)烷基,(C 2 -C 4)烯基,(C 1 -C 4)-环烷基; R 5是氢,(C 1 -C 4)烷基,(C 1 -C 4)链烯基,(C 1 -C 4)炔基,(C 1 -C 4)-环烷基,(C 1 -C 4)环烯基,(C 1 -C 4)-卤代烷基或(C 4)。 -C 5烷氧基(C 1 -C 4)烷基,X为氧,硫或-NR 3基团; R 5是氢,(C 1 -C 4)烷基,(C 1 -C 4)链烯基,(C 1 -C 4)炔基,(C 1 -C 4)-环烷基,(C 1 -C 4)环烯基,(C 1 -C 4)-卤代烷基或(C 4)。 -C 5烷氧基(C 1 -C 4)烷基是指并包括其生物学上可接受的酸加成盐。式I化合物是新颖的,并且也被本发明涵盖。

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