首页> 外国专利> CONDENSED DIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND METHODS CONTAINING THESE COMPOUNDS FOR THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM AND FOR THE PROMOTION OF CEREBRAL BLOODS

CONDENSED DIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND METHODS CONTAINING THESE COMPOUNDS FOR THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM AND FOR THE PROMOTION OF CEREBRAL BLOODS

机译:缩二氮杂酮,其制备方法和包含这些化合物的方法,用于治疗中枢神经系统疾病和促进脑血栓

摘要

The invention relates to novel condensed diazepinones of the general formula I IMAGE in which B represents one of the divalent radicals IMAGE and X, l, m, n and R1 to R7 are as defined in Claim 1, and in addition to their salts with inorganic or organic acids and a process for their preparation. The substances are used to improve or normalise disorders of cerebral perfusion due to arteriosclerosis, to treat diseases of the central nervous system, in particular Alzheimer's disease and Parkinson's disease, and as vagal pacemakers for the treatment of bradycardias and bradyarrhythmias, and also for improving memory power.
机译:本发明涉及通式I 的新型稠合二氮杂松酮,其中B代表二价基团之一,并且X,l,m,n和R 1至R 7如权利要求所定义。 1,它们与无机或有机酸形成的盐以及它们的制备方法。该物质用于改善或归因于动脉硬化的脑灌注紊乱,用于治疗中枢神经系统疾病,尤其是阿尔茨海默氏病和帕金森氏病,以及用于治疗心动过缓和心律过缓的迷走神经起搏器,以及用于改善记忆力功率。

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