首页> 外国专利> PROCESS FOR THE PREPARATION OF A MODIFIED LIPOPROTEIN BY INCORPORATION OF AN ACTIVE LIPOPHILIC SUBSTANCE, MODIFIED LIPOPROTEIN THUS OBTAINED AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING THE SAME.

PROCESS FOR THE PREPARATION OF A MODIFIED LIPOPROTEIN BY INCORPORATION OF AN ACTIVE LIPOPHILIC SUBSTANCE, MODIFIED LIPOPROTEIN THUS OBTAINED AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING THE SAME.

机译:通过掺入活性脂蛋白,从而获得修饰的脂蛋白的方法,所获得的脂蛋白被修饰并且包含相同的药物或化妆品组合物。

摘要

A method for preparing a lipoprotein modified by the incorporation of at least one lipophilic active substance other than a triglyceride, wherein said active substance is incorporated into an emulsion of a lipid phase in an aqueous continuous phase, an initial lipoprotein and at least one lipid transfer protein are stirred into the emulsion, the mixture is allowed to incubate, and the lipoprotein incorporating the active substance is isolated by known methods. The resulting modified lipoprotein, and a pharmaceutical or cosmetic composition containing said lipoprotein, are also described.
机译:一种制备通过掺入除甘油三酸酯以外的至少一种亲脂性活性物质修饰的脂蛋白的方法,其中将所述活性物质掺入水连续相的脂质相,初始脂蛋白和至少一种脂质转移的乳液中将蛋白搅拌到乳液中,使混合物温育,并通过已知方法分离掺入活性物质的脂蛋白。还描述了所得的修饰的脂蛋白,以及含有所述脂蛋白的药物或化妆品组合物。

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