首页> 外国专利> if etherifizierte or esterifizierte in position 2 substituted 4 - oh - chinolincarbonsaeurederivate, processes and intermediates for their preparation, their use as medicines and preparations containing them.

if etherifizierte or esterifizierte in position 2 substituted 4 - oh - chinolincarbonsaeurederivate, processes and intermediates for their preparation, their use as medicines and preparations containing them.

机译:如果位置2上的醚菲齐尔或酯菲齐尔取代了4-OH-chinolincarbonsaeurederivate,其制备方法和中间体,用作药物和包含它们的制剂。

摘要

Compounds of formula (I): IMAGE in which X at 5, 6, 7 or 8 is H, halogen, (C1-5) alkyl, (C1-4) alkoxy, -CF3, -SCF3, -OCF3, R1 is phenyl optionally substituted by at least OH, (C1-5) alkyl, (C1-4) alkoxy, CF3, NO2, halogen or a heterocyclic radical optionally substituted by a (C1-4) alkyl radical, R2 and R3 which are identical or different are H, (C1-4) alkyl, aryl, -C(:O)-R5, R5 being (C1-4) alkyl or aryl. R4 is H, (C1-4) alkyl or aryl, and their addition salts with acids and bases.
机译:式(I)的化合物:,其中在5、6、7或8处的X为H,卤素,(C1-5)烷基,(C1-4)烷氧基,-CF3,-SCF3,-OCF3,R1是任选至少被OH,(C1-5)烷基,(C1-4)烷氧基,CF3,NO2,卤素或任选被(C1-4)烷基取代的杂环基的苯基,R2和R3相同或不同的是H,(C 1-4)烷基,芳基,-C(∶O)-R 5,R 5为(C 1-4)烷基或芳基。 R 4是H,(C 1-4)烷基或芳基,以及它们与酸和碱的加成盐。

著录项

  • 公开/公告号AT87625T

    专利类型

  • 公开/公告日1993-04-15

    原文格式PDF

  • 申请/专利权人 ROUSSEL-UCLAF;

    申请/专利号AT19860401661T

  • 申请日1986-07-24

  • 分类号C07D417/12;C07D401/12;C07D413/12;C07D417/14;A61K31/47;A61K31/505;C07D215/56;C07D265/22;

  • 国家 AT

  • 入库时间 2022-08-22 05:09:25

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