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Pharmaceutical form consisting of a metered combination, for the treatment of premenopausal women.

机译:由计量组合组成的药物形式,用于治疗绝经前妇女。

摘要

Disclosed herein is a method of applying a HORMONE REPLACEMENT THERAPY AND BIRTH CONTROL A WOMAN premenopausal, comprising ADMINSTRAR premenopausal A WOMAN THAT NEED A combined dosage form of estrogen selected from 0.5-2.0 MG 17beta-estradiol, 0.008 to 0.030 mg ethinyl estradiol and mestranol 0.015 to 0.060 MG; AND BETWEEN SELECTED PROGETOGENO 0.025 to 0.100 mg levonorgestrel, 0.010-0, 070 MG OF gestodene, 0.025 to 0.100 mg desogestrel 0.025 to 0.100 mg 3-ketodesogestrel and 0.085 to 0.35 mg norethindrone, administered such an COMBINED DOSAGE for 23-25 ​​DAYS AND STARTING IN THE FIRST DAY OF MENSTRUAL CYCLE, FOLLOWED BY 2 TO 5 DAYS WITHOUT PILLS OR PLACEBO PILLS FOR A TOTAL OF 28 DAYS CYCLE MANAGEMENT'S. The dosage form FAVORITE invention is a combination of 1 mg 17beta-estradiol and 0.050 or 0.075 mg levonorgestrel. CYCLE MANAGEMENT OF THE INVENTION PREFERRED ADMINISTRATION OF COMBINED DOSAGE FORM DURING THE FIRST 24 DAYS OF ANY menstrual cycle and dosage form during the last 4 days of the menstrual cycle.
机译:本文公开了一种应用激素替代疗法和避孕方法来控制妇女绝经前的方法,其包括需要女性的联合剂型的雌激素的联合剂型,所述雌激素选自0.5-2.0 MG17β-雌二醇,0.008至0.030mg的乙炔基雌二醇和雌二醇0.015的联合剂型。到0.060 MG;以及在选定的PROGETOGENO 0.025至0.100 mg左炔诺孕酮,0.010-0、070 MG孕二烯酮,0.025至0.100 mg去氧孕烯0.025至0.100 mg 3-酮去孕孕酮和0.085至0.35 mg炔诺酮之间,以此类联合剂量给药23-25天并从月经周期的第一天开始,接着是2到5天,没有药丸或便药,总共进行了28天的周期管理。 FAVORITE发明的剂型是1mg17β-雌二醇和0.050或0.075mg左炔诺孕酮的组合。本发明的周期管理优选在任何月经周期的前24天期间管理联合剂型,并且在月经周期的后4天内对剂型进行管理。

著录项

  • 公开/公告号ES2033850T3

    专利类型

  • 公开/公告日1993-04-01

    原文格式PDF

  • 申请/专利权人 AMERICAN HOME PRODUCTS CORPORATION;

    申请/专利号ES19870306174T

  • 发明设计人 UPTON GERTRUDE VIRGINIA;

    申请日1987-07-13

  • 分类号A61K31/565;

  • 国家 ES

  • 入库时间 2022-08-22 05:09:01

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