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The piridobenzochiajin derivative null which has high anti-bacterial activity and the high biological utilization talent for
The piridobenzochiajin derivative null which has high anti-bacterial activity and the high biological utilization talent for
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机译:具有较高的抗菌活性和较高的生物利用才华的吡啶并苯并恶亚金衍生物无效
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摘要
Pyrido-benzothiazine derivatives having the following general formula: CHEM in which R is H or a C1-C6 alkyl or a C1-C6 fluoroalkyl, and R1 is N-alkyl-3-pyrrolidinalkylamine with C1 to C6 alkyls or CHEM where R2 is a C1-C6 alkyl or a C2-C6 alkenyl or an arylalkyl group, possibly substituted by halogen, hydroxy or keto-groups, both in the racemic form and in the optically active form. The invention also comprises the process for the preparation of derivatives of formula (I) starting from 2.4-difluoro-3-chloronitrobenzene. Said derivatives possess a high antibacterial acitvity as well as a high bioavailability to tissues; the invention also refers to pharmaceutical compositions containing them as active components.
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