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4- 3- Ethyl- 3- (propylsulfonyl) propyl amino -2-hydroxypropoxy benzonitrile stereoisomers yield and application

机译:4- [3- [乙基-[3-(丙基磺酰基)丙基]氨基] -2-羟基丙氧基]苄腈立体异构体的产量和应用

摘要

4-[3-[ethyl[3-((R*)-(propylsulfinyl)propyl]amino]-2(R)-hydroxypropoxy] -benzo n itrile, 4-[3-[ethyl[3-((S*)-(propylsulfinyl)propyl]amino]-2(R)-hydroxypropoxy] -benz on itrile, 4-[3-[ethyl[3-((R*)-(propylsulfinyl)propyl]amino]-2(S)-hydroxypropoxy] -benz on itrile, 4-[3-[ethyl[3-[((S*)-(propylsulfinyl)propyl]amino]-2(S)-hydroxypropoxy ]-ben zo nitrile and pharmaceutically acceptable salt thereof, processes for their preparation, as well as the use of said compounds for the preparation of medicaments with action against cardiac arrhythmias.
机译:4- [3- [乙基[3-((R *)-(丙基亚磺酰基)丙基]氨基] -2(R)-羟基丙氧基]-苯并-n,4,[3- [乙基[3-((S * )-(丙基亚硫酰基)丙基]氨基] -2(R)-羟基丙氧基]-苯并在4- [3- [乙基[3-((R *)-(丙基亚硫酰基)丙基]氨基] -2(S) -羟基上的-羟基丙氧基]-苯甲基,4- [3- [乙基[3-[((S *)-(丙基亚硫酰基)丙基]氨基] -2(S)-羟基丙氧基]-苯甲腈及其药学上可接受的盐,的制备方法,以及所述化合物在制备具有抗心律不齐作用的药物中的用途。

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