首页> 外国专利> DRUG FORMULATIONS COMPRISING COATED, VERY SPARINGLY WATER-SOLUBLE DRUGS FOR INHALATIONAL PHARMACEUTICAL FORMS, AND PROCESS FOR THEIR PREPARATION

DRUG FORMULATIONS COMPRISING COATED, VERY SPARINGLY WATER-SOLUBLE DRUGS FOR INHALATIONAL PHARMACEUTICAL FORMS, AND PROCESS FOR THEIR PREPARATION

机译:药物配方,包括用于药物制剂的包衣的,非常少量的水溶性药物及其制备方法

摘要

Drug formulations comprising coated, very sparingly water-soluble drugs for inhalational pharmaceutical forms, and process for their preparation Drug formulations comprising micronized particles of very sparingly water-soluble drugs which are coated with a natural, physiologically acceptable ampholytic surfactant soluble in water to give a micellar/colloidal solution, and a process for the preparation of these drug formulations, are described. When placed in an appropriate final container and after the addition of a chlorine-free, partially fluorinated propellant gas liquefiable under pressure, these formulations are suitable for inhalation.
机译:包含用于吸入药物形式的包衣的,非常少量的水溶性药物的药物制剂及其制备方法包含非常难溶于水的药物的微粉化颗粒的药物制剂,其被天然的,生理上可接受的溶于水的两性表面活性剂包被,得到描述了胶束/胶体溶液,以及这些药物制剂的制备方法。将这些制剂放在适当的最终容器中,并添加无氯的,部分氟化的,可在压力下液化的推进剂气体后,适合吸入。

著录项

  • 公开/公告号CA2128034A1

    专利类型

  • 公开/公告日1995-01-16

    原文格式PDF

  • 申请/专利权人 HOECHST AKTIENGESELLSCHAFT;

    申请/专利号CA19942128034

  • 发明设计人 REUL BERNHARD;PETRI WALTER;

    申请日1994-07-14

  • 分类号A61K9/12;A61K9/72;A61K31/34;A61K31/44;

  • 国家 CA

  • 入库时间 2022-08-22 04:16:13

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号