A novel human immunodeficiency virus (HIV) protease inhibitory compound having anti-AIDS effect and a method for producing the same

摘要

The present invention relates to an inhibitory compound of human immunodeficiency virus (HIV) protease represented by the following general formula (I), a process for producing the same, and a composition for the treatment or prevention of acquired immunodeficiency caused by HIV infection.;Wherein A is a functionalized acyl represented by the following general formula:;n is 0 or 1, R^One(C_OneTo C₄) Lower alkyl or amide substituted (C_OneTo C₂) Lower alkyl, R²Silver (C_OneTo C₄) Lower alkoxy, and an aromatic group containing a nitrogen atom, B is a functionalized amine represented by the following general formula (II);R³And R⁴Are each independently (C_OneTo C₄) Lower alkyl, an aromatic radical, an aromatic radical substituted with (C_OneTo C₄) Lower alkyl.