New benzo isoxazole and benzoisochiazoru chemical compound, the manufacturing method and medical supply constituent

摘要

New benzisoxazole and benzisothiazole derivatives usable as medication and corresponding to the formula: …IMAGE… in which: … …  - each of X1, X2, X3, X4 and X5, which are identical or different, is: hydrogen, halogen, [(C1-C5)-alkyl, -alkoxy or -alkylthio], hydroxyl, acyloxy, trifluoromethyl, nitro, amino or acetamido, or …  - two of them, in adjacent position, together form a methylenedioxy, ethylenedioxy or vinylenedioxy radical; …  - R1 is hydrogen or C1-C5 alkyl; …  - each of m and n denotes zero, one, two or three on condition that m + n is /= 1; …  - p is zero or an integer from 1 to 6; …  - q is two or three and …  - Y is oxygen or S(O)z, z being zero, one or two;… in racemic and optically active form. … …??These derivatives and their physiologically tolerable salts can be employed in therapeutics as sedative, anxiolytic, antiaggressive and analgesic agents and for the treatment of schizophrenia and of depression.