首页> 外国专利> N-ACYLPIPERIDINYLCARBONYLAMINOCARBOXYLIC ACIDS AND THEIR USE AS GLYCOPROTEIN IIB/IIIA ANTAGONISTS AND FIBRINOGEN-BLOOD PLATELETS BINDING INHIBITORS

N-ACYLPIPERIDINYLCARBONYLAMINOCARBOXYLIC ACIDS AND THEIR USE AS GLYCOPROTEIN IIB/IIIA ANTAGONISTS AND FIBRINOGEN-BLOOD PLATELETS BINDING INHIBITORS

机译:N-酰基哌啶基碳纳米管羧酸及其作为糖蛋白IIB / IIIA拮抗剂和血纤蛋白血血小板结合抑制剂

摘要

This invention relates to .beta.-alanine derivatives represented by formula(Ia) wherein each symbol is as defined in the specification andpharmaceutically acceptable salt thereof which is glycoprotein IIB/IIIaantagonist, inhibitor of blood platelets aggregation and inhibitor of thebinding of fibrinogen to blood platelets, to processes for the preparationthereof, to a pharmaceutical composition comprising the same and to a methodfor the prevention and/or treatment diseases indicated in the specification toa human being or an animal.
机译:本发明涉及由下式表示的β-丙氨酸衍生物(Ia)其中每个符号如说明书中所定义,并且其药学上可接受的盐是糖蛋白IIB / IIIa拮抗剂,血小板凝集抑制剂及其抑制剂纤维蛋白原与血小板的结合,以及制备过程其,包含其的药物组合物和方法用于规范中指出的预防和/或治疗疾病人类或动物。

著录项

  • 公开/公告号CA2215106A1

    专利类型

  • 公开/公告日1996-09-26

    原文格式PDF

  • 申请/专利权人 FUJISAWA PHARMACEUTICAL CO. LTD.;

    申请/专利号CA19962215106

  • 申请日1996-03-14

  • 分类号C07D211/60;C07D471/04;C07D401/06;C07F7/10;C07D401/14;C07D405/14;C07D409/14;C07D411/14;C07D413/14;C07D417/14;C07D217/26;A61K31/435;A61K31/495;A61K31/535;A61K31/54;A61K31/695;

  • 国家 CA

  • 入库时间 2022-08-22 03:50:12

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