首页> 外国专利> (R)-4-(2-(3-CYCLOPENTYLOXY-4-METHOXYPHENYL)-2-PHENYLETHYL) PYRIDINE HYDROGEN SULPHATE SALT AS PDE TYPE IV INHIBITOR

(R)-4-(2-(3-CYCLOPENTYLOXY-4-METHOXYPHENYL)-2-PHENYLETHYL) PYRIDINE HYDROGEN SULPHATE SALT AS PDE TYPE IV INHIBITOR

机译：（R）-4-（2-（3-（3-环戊氧基-4-甲氧基苯基）-2-苯基乙基）吡啶硫酸氢盐作为PDE IV型抑制剂

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摘要

The hydrogen sulphate salt of the selective phosphodiesterase type IV inhibitor (R)-4-[2-(3-Cyclopentyloxy-4-methoxyphenyl)-2-phenylethyl]- pyridine hydrogen sulphate salt is described. The salt possesses a number of advantageous chemical and physical characteristics making it particularly suitable for pharmaceutical formulation for use in inter alia the prophylaxis and treatment of asthma.

机译：描述了选择性磷酸二酯酶IV型抑制剂（R）-4- [2-（3-环戊氧基-4-甲氧基苯基）-2-苯基乙基]-吡啶硫酸氢盐的硫酸氢盐。该盐具有许多有利的化学和物理特性，使其特别适合用于尤其是预防和治疗哮喘的药物制剂。

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公开/公告号WO9535282A1

专利类型
公开/公告日1995-12-28

原文格式PDF
申请/专利权人 CELLTECH THERAPEUTICS LIMITED;
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申请/专利号WO1995GB01460
发明设计人 WARRELLOW GRAHAM JOHN;HEAD JOHN CLIFFORD;BOYD EWAN CAMPBELL;ALEXANDER RIKKI PETER;
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申请日1995-06-21
分类号C07D213/30;A61K31/44;
国家 WO
入库时间 2022-08-22 03:49:13

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