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Medicament for treating or preventing cerebrovascular disease (medicament for treating or preventing cerebrovascular diseases)

机译:治疗或预防脑血管疾病的药物(治疗或预防脑血管疾病的药物)

摘要

The present invention relates to the use of a compound of the following general formula (I), (II) or (III) or a pharmaceutically acceptable salt thereof for the preparation of a medicament for the treatment or prophylaxis of cerebrovascular diseases:;Wherein ROneIs hydrogen, lower alkyl, lower alkenyl or N, N-di (lower) alkylaminomethyl, R2Is hydrogen, lower alkyl or halogen and R3Is imidazolyl or pyridyl, each of which may have suitable substituent (s) and R4Is hydrogen, lower alkyl, lower alkenyl or hydroxy (lower) alkyl, R5Is hydrogen, hydroxy or acyloxy, or R4And R5Are joined together to form an additional bond, R6, R7And R8Are each hydrogen, lower alkyl, lower alkenyl, aryl or ar (lower) alkyl, R9Is imidazolyl, or pyridyl, which may have suitable substituent (s), A is lower alkylene, Is a single bond or a double bond.
机译:本发明涉及以下通式(I),(II)或(III)的化合物或其药学上可接受的盐在制备用于治疗或预防脑血管疾病的药物中的用途: 一个是氢,低级烷基,低级烯基或N,N-二(低级)烷基氨基甲基,R 2 是氢,低级烷基或卤素和R 3 < / Sup>是咪唑基或吡啶基,它们各自可以具有合适的取代基,R 4 是氢,低级烷基,低级烯基或羟基(低级)烷基,R 5 是氢,羟基或酰氧基,或R 4 和R 5 连接在一起形成另一个键R 6 ,R < Sup> 7 和R 8 分别是氢,低级烷基,低级烯基,芳基或芳基(低级)烷基,R 9 是咪唑基或吡啶基,可以具有合适的取代基的化合物,A是低级亚烷基,是单键或双键。

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