where 1m represents imidazole group having formula , R1 represents atom of hydrogen or C1-4 alkyl, C3-4 alkenyl, C3-4 alkynyl, C5-6 cycloalkyl, C5-6 cycloalkylmethyl, benzyl, phenylmethoxymethyl or N,N-diC1-3 alkylcarboxamino group. EFFECT: improves quality of desired product. 1 tbl"/> DERIVATIVES OF LACTAM AND PHARMACEUTICAL COMPOSITION BEING ANTAGONIST OF 5-OXYTRAPTAMINE(5-HT) FOR 5-HT<Sub>3</Sub> RECEPTORS OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS AND SOLVATES
首页> 外国专利> DERIVATIVES OF LACTAM AND PHARMACEUTICAL COMPOSITION BEING ANTAGONIST OF 5-OXYTRAPTAMINE(5-HT) FOR 5-HT3 RECEPTORS OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS AND SOLVATES

DERIVATIVES OF LACTAM AND PHARMACEUTICAL COMPOSITION BEING ANTAGONIST OF 5-OXYTRAPTAMINE(5-HT) FOR 5-HT3 RECEPTORS OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS AND SOLVATES

机译:内酰胺和药物成分的衍生物为5-羟色胺(5-HT)对5-HT 3 受体或它们的可药用盐和溶剂的拮抗剂

摘要

FIELD: organic chemistry, medicine. SUBSTANCE: desired compounds have common formula where 1m represents imidazole group having formula , R1 represents atom of hydrogen or C1-4 alkyl, C3-4 alkenyl, C3-4 alkynyl, C5-6 cycloalkyl, C5-6 cycloalkylmethyl, benzyl, phenylmethoxymethyl or N,N-diC1-3 alkylcarboxamino group. EFFECT: improves quality of desired product. 1 tbl
机译:领域:有机化学,医学。物质:所需化合物具有通用公式,其中1m代表咪唑基具有公式,R 1 表示氢或C 1-4 烷基,C 3-4 烯基,C 3-4 炔基,C 5-的原子6 环烷基,C 5-6 环烷基甲基,苄基,苯甲氧基甲基或N,N-diC 1-3 烷基羧氨基。效果:提高所需产品的质量。 1汤匙

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