首页> 外国专利> DIAMIDES OF MIXED PIRIDINE-2,4- AND -2,5-DICARBOXYL ACIDS, PROCEDURE FOR THEIR PREPARATION, USE OF THE SAME, AS WELL AS DRUGS BASED ON THESE COMPOUNDS.

DIAMIDES OF MIXED PIRIDINE-2,4- AND -2,5-DICARBOXYL ACIDS, PROCEDURE FOR THEIR PREPARATION, USE OF THE SAME, AS WELL AS DRUGS BASED ON THESE COMPOUNDS.

机译:混合吡啶-2,4-和-2,5-二羧酸的二酰胺,其制备方法,使用相同的方法以及基于这些化合物的药物。

摘要

THE INVENTION CONCERNS MIXED DIAMIDES OF 2,4,5-PIRIDINDICARBOXILICO ACID, WHERE THE AMIDA GROUP OF CARBOXILICO ACID IN POSITION 2 REPRESENTS A PRIMARY ACID AMIDA. THE MENTIONED COMPOUNDS ARE SUITABLE FOR INHIBITION OF PROLINHYDROXYLASE AND LYSINHYDROXYLASE AND ARE USED AS FIBROSUPPRESSANTS AND IMMUNOSUPPRESSANTS.
机译:本发明涉及2,4,5-吡啶二羧酸羧酸的混合二胺,其中位置2的羧酰胺的酰胺基团代表主要的酸酰胺。所述的化合物适合于抑制脯氨酰羟化酶和赖氨酰羟化酶,并用作纤维抑制剂和免疫抑制剂。

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