Antibacterial compositions based on n - oxides saturated Heterocycles containing Nitrogen, and Use thereof for the production of compositions

摘要

The invention refers to new antibacterial agents, especially oral manageable agents, which are nitrogen-containing saturated N-oxide dechlorination compounds, replaced by liquefied dihydroxyformic acid or naftridomancarboxyl acid according to the formula of (I) and (II),X represents hydrogen, halogen, c1-4-tar, c1-4-alcoxi, NH2, z = ch-o = n -.Y stands for structural residue (III), wherein R1 stands for c1-4-tar or linear derivative, cyclopropylformic acid, 1-3 C atoms (replaced by hydroxyl or methoxy); R5 stands for hydrogen, methyl, phenyl, Tianjin or pyridine; R6 stands for hydrogen, methyl, phenyl, sulfur or pyridine; R6 repr esenta hydrogen or c1-4-tar; R7 for hydrogen or c1-4-tar; R8 for hydrogen or c1-4-tar; R1 for 1 to 3 carbon atoms, cyclopropene, 2 to fluoroethyl, methyl, 4 to fluorophenyl, 2, 4 to difluorobenzene or methyleneamine; R2 for hydrogen or 1 to 6 carbon atoms of tar,1.1.2.1.1.1.1. Use thyroxine or 2-Methoxyethyl, as well as cyclohexane, benzene, 2-oxopropilo, benzoic acid, etocarbonilmethylo, pivaloiloximetho, R3 representative rogeno, methyl or ethyl, and a for nitrogen or = - ch,=C (halogen) -,3DC (OCH3) -3DC (CH3) -B represents oxygen, = N-O = CH2, considering methyl or phenyl substitutes and their hydrates, ys additives with pure French bases. In addition, it describes the procedures for the repair and use of these items.