首页> 外国专利> PROCESS FOR PRODUCING STABILE AQUOUS COMPOSITIONS CONTAINING 5,10-METHYLENE-TETRAHYDRO-FOLIC ACID AND PROCESS FOR PRODUCING 5,10-METHYLENE-TETRAHYDRO-FOLIC ACID/CYCLODEXTRIN INCLUSION COMPOUNDS

PROCESS FOR PRODUCING STABILE AQUOUS COMPOSITIONS CONTAINING 5,10-METHYLENE-TETRAHYDRO-FOLIC ACID AND PROCESS FOR PRODUCING 5,10-METHYLENE-TETRAHYDRO-FOLIC ACID/CYCLODEXTRIN INCLUSION COMPOUNDS

机译:包含5,10-亚甲基-四氢叶酸的稳定水溶液成分的制备方法及包含5,10-亚甲基-四氢叶酸/环糊精的化合物的制备步骤

摘要

The invention relates to cyclodextrin inclusion compounds of 5,10-methylenetetrahydrofolic acid. The surprisingly high stability of these compounds makes it possible to use them pharmaceutically for the first time. The invention also relates to a process for preparing the said substances and to their use for producing pharmaceutical compositions.
机译:本发明涉及5,10-亚甲基四氢叶酸的环糊精包合物。这些化合物的惊人的高稳定性使其首次可药用。本发明还涉及制备所述物质的方法及其在制备药物组合物中的用途。

著录项

  • 公开/公告号NO303715B1

    专利类型

  • 公开/公告日1998-08-24

    原文格式PDF

  • 申请/专利权人 EPROVA AG;

    申请/专利号NO19930002517

  • 申请日1993-07-09

  • 分类号A61K31/505;A61K47/40;C07D475/04;

  • 国家 NO

  • 入库时间 2022-08-22 02:57:12

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